General Information of This Peptide
Peptide ID
BTDP008704
Peptide Name
Potassium channel toxin alpha-KTx 6.15
Symonym
Hemitoxin
Species
Hemiscorpius lepturus (Scorpion)
Uniprot Name
KAX6F_HEMLE
Alphafold ID
P85528
3D Structure
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2D Sequence
3D Structure
Source
Alphafold db: P85528
Sequence
IKCTLSKDCYSPCKKETGCPRAKCINRNCKCYGCS
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Sequence Length
35
Mass (Da)
3906
Sequence Removed Signal Peptide
IKCTLSKDCYSPCKKETGCPRAKCINRNCKCYGCS
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Disulfide Bond
3-24;9-29;13-31;19-34
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Kingdom: Metazoa
Phylum: Arthropoda
Class: Arachnida
Order: Scorpiones
Family: Hemiscorpiidae
Genus: Hemiscorpius
Species: Hemiscorpius lepturus
Full List of Activity Data of This Peptide Toxin
                        Target Name Activity Data Type Activity Data Concentration Note Reference
 Target Info    Kv1.3 IC50
2 nM
.
Blocker
[1]
 Target Info    Kv1.3 IC50
2 nM
.
Blocker
[1]
 Target Info    Kv1 IC50
13 nM
.
Blocker
[1]
 Target Info    Kv1 IC50
13 nM
.
Blocker
[1]
 Target Info    Kv1 IC50
16 nM
.
Blocker
[1]
 Target Info    Kv1.2 IC50
16 nM
.
Blocker
[1]
 Target Info    Kv1.2 IC50
16 nM
.
Blocker
[1]
References
Ref 1 Hemitoxin, the first potassium channel toxin from the venom of the Iranian scorpion Hemiscorpius lepturus. FEBS J. 2008 Sep;275(18):4641-50. doi: 10.1111/j.1742-4658.2008.06607.x. Epub 2008 Aug 11.
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