General Information of This Peptide
Peptide ID
BTDP005618
Peptide Name
[des-Arg1]-proctolin
Symonym
NEP-inhibiting peptide
Species
Tityus serrulatus (Brazilian scorpion)
Uniprot Name
PRCT_TITSE
3D Structure
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2D Sequence
3D Structure
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Predict by Alphafold2
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Alphafold Parameters: msa_mode: mmseqs2_uniref_env model_type: auto num_recycles: auto
Sequence
YLPT
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Sequence Length
4
Mass (Da)
493
Sequence Removed Signal Peptide
YLPT
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        Click to Show/Hide the Complete Species Lineage
Kingdom: Metazoa
Phylum: Arthropoda
Class: Arachnida
Order: Scorpiones
Family: Buthidae
Genus: Tityus
Species: Tityus serrulatus
Full List of Activity Data of This Peptide Toxin
                        Target Name Activity Data Type Activity Data Concentration Note Reference
 Target Info    peptidase neprilysin (NEP/MME) Inhibition constant
0.94 μM
. . [1]
 Target Info    endopeptidase EP24.15 Inhibition constant
36 μM
. . [1]
 Target Info    endopeptidase EP24.15 Inhibition constant
74 μM
. . [1]
References
Ref 1 [des-Arg(1)]-Proctolin: A novel NEP-like enzyme inhibitor identified in Tityus serrulatus venom. Peptides. 2016 Jun;80:18-24. doi: 10.1016/j.peptides.2015.05.013. Epub 2015 Jun 6.
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