General Information of This Peptide
Peptide ID
BTDP000478
Peptide Name
Potassium channel toxin ShK (M21M[Dap])
Symonym
Potassium channel toxin ShK (M21M[Dap])
3D Structure
Original Sequence
RSCIDTIPKSRCTAFQCKHSMKYRLSFCRKTCGTC
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Mutant Sequence
RSCIDTIPKSRCTAFQCKHSM[Dap]YRLSFCRKTCGTC
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Sequence Length
35
Mass(Da)
4013
Sequence Removed Signal Peptide
RSCIDTIPKSRCTAFQCKHSM[Dap]YRLSFCRKTCGTC
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PDB ID
1BEI
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N.A.
Full List of Activity Data of This Peptide Toxin
                        Target Name Activity Data Type Activity Data Concentration Note Reference
 Target Info    Kv1.5 Inhibition rate .
100 nM
Blocker
[1]
 Target Info    KCa4 Inhibition rate .
100 nM
Blocker
[1]
References
Ref 1 ShK-Dap22, a potent Kv1.3-specific immunosuppressive polypeptide. J Biol Chem. 1998 Dec 4;273(49):32697-707. doi: 10.1074/jbc.273.49.32697.
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